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William R Roeske Selected Research

methyl- 2',6'- dimethyltyrosinyltetrahydroisoquinoline- 3- carboxylic acid

2/2003(2S,3R) beta-methyl-2',6'-dimethyltyrosine-L-tetrahydroisoquinoline-3-carboxylic acid [(2S,3R)TMT-L-Tic-OH] is a potent, selective delta-opioid receptor antagonist in mouse brain.

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William R Roeske Research Topics

Disease

8Pain (Aches)
06/2012 - 12/2003
6Hyperalgesia
06/2012 - 12/2008
1Ischemia
07/2007
1Myocardial Infarction
07/2007
1Infarction (Infarctions)
07/2007
1Myocardial Ischemia (Ischemic Heart Diseases)
07/2007
1Chronic Pain
07/2006
1Tics (Tic)
02/2003

Drug/Important Bio-Agent (IBA)

7Opioid Analgesics (Opioids)IBA
06/2012 - 12/2003
6Morphine (MS Contin)FDA LinkGeneric
06/2012 - 07/2006
6Neurotransmitter Agents (Neurotransmitter)IBA
12/2010 - 12/2003
5Calcitonin Gene-Related PeptideIBA
12/2010 - 04/2008
2Analgesics (Analgesic Drugs)IBA
04/2008 - 07/2006
2delta Opioid Receptors (delta Opioid Receptor)IBA
07/2007 - 02/2003
1Tryptophan (L-Tryptophan)FDA Link
06/2012
1Neurokinin-1 Receptors (Neurokinin 1 Receptor)IBA
06/2012
1TachykininsIBA
06/2012
1Pharmaceutical PreparationsIBA
06/2012
1AM 1241IBA
03/2012
1Cannabinoid Receptors (Cannabinoid Receptor)IBA
03/2012
1Cyclic AMP (AMP, Cyclic)IBA
12/2010
1ProstaglandinsIBA
12/2010
1Cyclic AMP-Dependent Protein Kinases (cAMP-Dependent Protein Kinase)IBA
12/2010
1Capsaicin (Zostrix)FDA Link
09/2009
1CannabinoidsIBA
05/2009
1Small Interfering RNA (siRNA)IBA
12/2008
15- iodo- 3- ((3,5- dibromo- 4- hydroxyphenyl)methylene)- 2- indolinoneIBA
04/2008
1Epinephrine (Adrenaline)FDA LinkGeneric
07/2007
1D-Penicillamine (2,5)- EnkephalinIBA
07/2007
1Opioid Peptides (Opioid Peptide)IBA
02/2003
1AcidsIBA
02/2003
1methyl- 2',6'- dimethyltyrosinyltetrahydroisoquinoline- 3- carboxylic acidIBA
02/2003
1hydroxide ionIBA
02/2003

Therapy/Procedure

1Analgesia
12/2003